2-chloroadenosine | Ligand Activity Charts | IUPHAR/BPS Guide to PHARMACOLOGY
2-chloroadenosine [Ligand Id: 372] activity data from GtoPdb and ChEMBL. Click here for a description of the charts and data ... ChEMBL ligand: CHEMBL285819 (2-Chloroadenosine) *A1 receptor/Adenosine A1 receptor in Human [ChEMBL: CHEMBL226] [GtoPdb: 18] [ ... Antagonism of cyclic [3H]AMP accumulation elicited by 15 uM 2-chloroadenosine in [3H]adenine-labeled guinea pig cerebral ...
2-Chloroadenosine - P. D. POLYCHEM PVT. LTD
The influence of 2‐chloroadenosine on potassium‐evoked and neurally‐evoked acetylcholine secretion from normal or from latent...
... chloroadenosine on potassium‐evoked and neurally‐evoked acetylcholine secretion from normal or from latent active zones in the ... chloroadenosine on potassium‐evoked and neurally‐evoked acetylcholine secretion from normal or from latent active zones in the ... Dive into the research topics of The influence of 2‐ ...
Erowid.org: Erowid Reference 3782 : Selectivity of cyproheptadine as assessed by radioligand binding : Williams M, Martin GE
5HT-2 ([3H]mianserin; rat forebrain; 0.75 nM; Peroutka & Snyder 1981); 5-HT-1 and 2 ([3H]lysergic acid diethylamide (LSD); 2 nM ... 5-HT-2 and muscarinic cholinergic receptor sites than in inhibiting depolarization dependent calcium fluxes (Donatsch et al ... 2-CADO; 1.0 nM; whole brain crude synaptic membranes; Williams & Risley 1980). Examination of cyproheptadine in eleven receptor ...
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Evidence for the presence of A1 adenosine receptors in the aorta of spontaneously hypertensive rats, NC DOCKS (North Carolina...
2 In phenylephrine contracted aortic rings concentration-response curves were constructed by cumulative additions (10711 ±1075 ... The contractile response in SHR was abolished by A1 adenosine receptor antagonist N6- endonorbornan-2-yl-9-methyladenine (N- ... 2-p-(-2-carboxyethyl) phenethylamino-5-N-thylcarboxamido adenosine (CGS-21680). 3 A non-speci®c adenosine receptor agonist 2- ... chloroadenosine (CAD) resulted in biphasic response with a small contraction at lower concentrations (1079 ±1078 M) followed ...
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Effect of metabolic products of muscular contraction on discharge of group III and IV afferents<...
Likewise, monobasic sodium phosphate (20 and 400 mM; 1 ml) and 2-chloroadenosine (50-100 μg) had only trivial effects on the ... Likewise, monobasic sodium phosphate (20 and 400 mM; 1 ml) and 2-chloroadenosine (50-100 μg) had only trivial effects on the ... Likewise, monobasic sodium phosphate (20 and 400 mM; 1 ml) and 2-chloroadenosine (50-100 μg) had only trivial effects on the ... Likewise, monobasic sodium phosphate (20 and 400 mM; 1 ml) and 2-chloroadenosine (50-100 μg) had only trivial effects on the ...
Dipyridamole. Medical search. Definitions
2-Chloroadenosine. A metabolically stable analog of adenosine which acts as an adenosine receptor agonist. The compound has a ... Equilibrative-Nucleoside Transporter 2. A subtype of equilibrative nucleoside transporter proteins that is insensitive to ... DipyridamoleDilazepAdenosineVasodilator AgentsThioinosineThallium RadioisotopesEquilibrative-Nucleoside Transporter 2 ... unlike positron-emission tomography where the positron-electron annihilation results in the emission of 2 photons at 180 ...
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Volume: 2 Issue: 3 Year: 2005 Page: 261-267. Author(s): Barney E. Dwyer, Atsushi Takeda, Xiongwei Zhu, George Perry, Mark A. ... Volume: 5 Issue: 2 Year: 2005 Page: 85-102. Author(s): Chung Fai Wong, Alexander Guminski, Nicholas A. Saunders, Andrew J. ... Volume: 1 Issue: 2 Year: 2005 Page: 157-166. Author(s): Yasuhiro Ito ... Cytostatic Effect of the Nucleoside Analogue 2-Chloroadenosine on Human Prostate Cancer Cell Line. Journal: Current ...
Chemistry and Biochemistry - Scholarly Works - University of Arizona
Weyand, N. J., Calton, C. M., Higashi, D. L., Kanack, K. J. & So, M., Jan 15 2010, In: Journal of Immunology. 184, 2, p. 694- ... Kondrashov, D. A., Roberts, S. A., Weichsel, A. & Montfort, W. R., Nov 2 2004, In: Biochemistry. 43, 43, p. 13637-13647 11 p.. ... Dietrich, M., Mollenkopf, H., So, M. & Friedrich, A., Jul 2009, In: FEMS Microbiology Letters. 296, 2, p. 248-256 9 p.. ... Harth, G., Haidaris, C. G. & So, M., Mar 1 1989, In: Molecular and Biochemical Parasitology. 33, 2, p. 143-150 8 p.. Research ...
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Adenosine - ADxS.org
2-chloroadenosine (CAD) is a non-specific adenosine receptor agonist62 3.6.2. Antagonists¶. *Xanthine *Caffeine (A2A and A1 ... 3.1.2. Effect mediated by A1 receptors¶. 3.1.2.1. Neurophysiological effect in the brain¶. * Inhibition of the release of ... 3.1.2. Effect mediated by A2A receptors¶. 3.1.2.1. Neurophysiological effect in the brain of A2A¶. *Reduction of dopamine D2 ... 4.1.2. Adenosine and adenosine antagonists inhibit D2 receptors in A2A-D2 heteromers¶. A2A-D2 heteromers occur primarily in the ...
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2. Gender Differences in the Circadian and Seasonal Variations in Patients with Takotsubo Syndrome: A Multicenter Registry at ... The average postoperative opacification rate in the first case was 7.36 + 1.12 (n = 2) in the RCA, 3.81 + 0.51 (n = 3) in the ... The patency rates of device-dependent SVGs that were 1, 2, 3, 4, 5, 6, 7, and 8 years old were 90.1% ± 1.8%, 87.1% ± 2.3%, 86.1 ... We recently encountered 2 patients with mobile cardiac calcified amorphous tumors who were successfully treated by surgery. ...
CERUTI, STEFANIA MARIA
2-Chloro-adenosine-induced apoptosis in rat brain neuron-glia primary cultures 1-gen-1995 S. CerutiF. CattabeniG. BurnstockD. ... 2-chloro-adenosine induces a glutamate-dependent calcium response in C2C12 myotubes 1-gen-2000 C. FrankA. GiammarioliL. Falzano ... A novel gliotic P2 receptor mediating cyclooxygenase-2 induction in rat and human astrocytes 1-gen-2000 R. BrambillaS. CerutiW ... 2-Chloro-adenosine-induced apoptosis in rat brain neuron-glia primary cultures. 1995 S. Ceruti, F. Cattabeni, G. Burnstock, D. ...
Science of Synthesis: Best methods. Best results - Thieme Chemistry
However, the direct preparation of 8-chloroadenosine and of its mono- and diphosphate derivatives can be achieved by using ... This method may be a convenient way to prepare N6-methyl derivatives of 8-chloroadenosine (78% yield).[325] ... An analogous chlorination (t-BuOCl, DMF, −70°C, 2 h) of 6-(methylamino)- and 6-(dimethylamino)purine nucleosides gives the ...
Adenosine production by human B cells and B cell-mediated suppression of activated T cells | Blood | American Society of...
For example, coculturing of CD19+ human B cells with CD4+CD25+ alloreactive T cells in the presence of IL-2 and CD28-specific ... 2-chloroadenosine (CADO) was purchased from Sigma-Aldrich and used in place of ADO, because of its greater stability. The ... C) The MFI values for surface expression of the 2 ectonucleotidases are higher in B cells than CD4+ T cells. Data are means ± ... C) The MFI values for surface expression of the 2 ectonucleotidases are higher in B cells than CD4+ T cells. Data are means ± ...
Deoxyadenosines | Profiles RNS
On the other hand, S228 displayed an upregulation in its phosphorylation level in response towards the Ca2+ switch by 1 - An...
Cells had been incubated in principal antibody diluted 2-Chloroadenosine (CADO) 1:100 in GSDB for 1 h at area temperature and ... Hence, the mRNA levels of integrin 1, integrin 2, integrin 1, RANKL and ALP mRNA in GroEL-stimulated PDL cells was analyzed ... 0.26 2-Chloroadenosine (CADO) M of every primer, and 2.5 units of Pfu turbo enzyme in 50 l. The mix was warmed at 95C for 2 min ... 2 mM l-glutamine, 50 U/mL penicillin, and 50 mg/mL streptomycin for 16 h. Cells had been then returned on track Ca2+-filled ...
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MH DELETED MN ADDED MN
ELAV-Like Protein 2 D12.776.641.520.500 D12.776.631.520.500 ELAV-Like Protein 3 D12.776.641.520.750 D12.776.631.520.750 ELAV- ... 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine D3.438.79.800 D3.633.100.79.800 2-Aminopurine D3.438.759.138.50 ... quinolizin-2-ol, 2-Ethyl-1,3,4,6,7,11b-hexahydro-3-isobutyl-9,10-dimethoxy- D3.438.834.700 D3.633.100.834.700 4- ... Ataxin-2 D12.776.641.69.750 D12.776.631.69.750 Ataxin-3 D8.811.277.656.300.887.500 D8.811.37.250 D12.776.641.69.875 D12.776. ...
MH DELETED MN ADDED MN
ELAV-Like Protein 2 D12.776.641.520.500 D12.776.631.520.500 ELAV-Like Protein 3 D12.776.641.520.750 D12.776.631.520.750 ELAV- ... 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine D3.438.79.800 D3.633.100.79.800 2-Aminopurine D3.438.759.138.50 ... quinolizin-2-ol, 2-Ethyl-1,3,4,6,7,11b-hexahydro-3-isobutyl-9,10-dimethoxy- D3.438.834.700 D3.633.100.834.700 4- ... Ataxin-2 D12.776.641.69.750 D12.776.631.69.750 Ataxin-3 D8.811.277.656.300.887.500 D8.811.37.250 D12.776.641.69.875 D12.776. ...
MH DELETED MN ADDED MN
ELAV-Like Protein 2 D12.776.641.520.500 D12.776.631.520.500 ELAV-Like Protein 3 D12.776.641.520.750 D12.776.631.520.750 ELAV- ... 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine D3.438.79.800 D3.633.100.79.800 2-Aminopurine D3.438.759.138.50 ... quinolizin-2-ol, 2-Ethyl-1,3,4,6,7,11b-hexahydro-3-isobutyl-9,10-dimethoxy- D3.438.834.700 D3.633.100.834.700 4- ... Ataxin-2 D12.776.641.69.750 D12.776.631.69.750 Ataxin-3 D8.811.277.656.300.887.500 D8.811.37.250 D12.776.641.69.875 D12.776. ...
MH DELETED MN ADDED MN
ELAV-Like Protein 2 D12.776.641.520.500 D12.776.631.520.500 ELAV-Like Protein 3 D12.776.641.520.750 D12.776.631.520.750 ELAV- ... 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine D3.438.79.800 D3.633.100.79.800 2-Aminopurine D3.438.759.138.50 ... quinolizin-2-ol, 2-Ethyl-1,3,4,6,7,11b-hexahydro-3-isobutyl-9,10-dimethoxy- D3.438.834.700 D3.633.100.834.700 4- ... Ataxin-2 D12.776.641.69.750 D12.776.631.69.750 Ataxin-3 D8.811.277.656.300.887.500 D8.811.37.250 D12.776.641.69.875 D12.776. ...
MH DELETED MN ADDED MN
ELAV-Like Protein 2 D12.776.641.520.500 D12.776.631.520.500 ELAV-Like Protein 3 D12.776.641.520.750 D12.776.631.520.750 ELAV- ... 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine D3.438.79.800 D3.633.100.79.800 2-Aminopurine D3.438.759.138.50 ... quinolizin-2-ol, 2-Ethyl-1,3,4,6,7,11b-hexahydro-3-isobutyl-9,10-dimethoxy- D3.438.834.700 D3.633.100.834.700 4- ... Ataxin-2 D12.776.641.69.750 D12.776.631.69.750 Ataxin-3 D8.811.277.656.300.887.500 D8.811.37.250 D12.776.641.69.875 D12.776. ...
DeCS 2009 - February 20, 2009 version
2-Fluoro-2-deoxyglucose use Fluorodeoxyglucose F18 2H-Benzo(a)quinolizin-2-ol, 2-Ethyl-1,3,4,6,7,11b-hexahydro-3-isobutyl-9,10- ... 2-Amino-5-phosphonovaleric Acid use 2-Amino-5-phosphonovalerate 2-Amino-6-(1,2,3-trihydroxypropyl)-4(3H)-pteridinone use ... 2-Oxoisovalerate Dehydrogenase (Lipoamide) use 3-Methyl-2-Oxobutanoate Dehydrogenase (Lipoamide) 2-PAM Compounds use ... 2-Chloroethyl Alcohol use Ethylene Chlorohydrin 2-Dehydro-3-Deoxyphosphoheptonate Aldolase use 3-Deoxy-7-Phosphoheptulonate ...
DeCS 2009 - February 20, 2009 version
2-Fluoro-2-deoxyglucose use Fluorodeoxyglucose F18 2H-Benzo(a)quinolizin-2-ol, 2-Ethyl-1,3,4,6,7,11b-hexahydro-3-isobutyl-9,10- ... 2-Amino-5-phosphonovaleric Acid use 2-Amino-5-phosphonovalerate 2-Amino-6-(1,2,3-trihydroxypropyl)-4(3H)-pteridinone use ... 2-Oxoisovalerate Dehydrogenase (Lipoamide) use 3-Methyl-2-Oxobutanoate Dehydrogenase (Lipoamide) 2-PAM Compounds use ... 2-Chloroethyl Alcohol use Ethylene Chlorohydrin 2-Dehydro-3-Deoxyphosphoheptonate Aldolase use 3-Deoxy-7-Phosphoheptulonate ...