![4-Amino-6-benzylamino-1,2-dihydro-2-phenyl-1,2,4-triazolo [4,3-alpha]-quinoxalin-1-one: a new A2A adenosine receptor antagonist...](data:image/png;base64,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)
4-Amino-6-benzylamino-1,2-dihydro-2-phenyl-1,2,4-triazolo [4,3-alpha]-quinoxalin-1-one: a new A2A adenosine receptor antagonist...
Novel human adenosine receptor antagonists based on the 7-amino-thiazolo[5,4-d]pyrimidine scaffold. Structural investigations...
The synthesized compounds 2-27 were evaluated in radioligand binding (A1, A2A and A3) and adenylyl cyclase activity (A2B and ... Novel human adenosine receptor antagonists based on the 7-amino-thiazolo[5,4-d]pyrimidine scaffold. Structural investigations ... Novel human adenosine receptor antagonists based on the 7-amino-thiazolo[5,4-d]pyrimidine scaffold. Structural investigations ... in order to evaluate their affinity and potency at human adenosine receptor subtypes. The current study allowed us to support ...
Recettori per l'adenosina - Wikipedia
Kalda A, Yu L, Oztas E, Chen JF, Novel neuroprotection by caffeine and adenosine A(2A) receptor antagonists in animal models of ... Lo stesso argomento in dettaglio: Recettore A1 per ladenosina. il recettore A1 è distribuito in tutto lorganismo. Questo ... Baraldi PG, Tabrizi MA, Gessi S, Borea PA, Adenosine receptor antagonists: translating medicinal chemistry and pharmacology ... Entrez Gene: ADORA2A adenosine A2A receptor, su ncbi.nlm.nih.gov. Jacobson KA, Gao ZG, Adenosine receptors as therapeutic ...
Exploring the QSAR of pyrazolo[3,4-b]pyridine, pyrazolo[3,4-b]pyridone and pyrazolo[3,4-b]pyrimidine derivatives as antagonists...
Pyrazolo[3,4-b]pyridines have been recently presented as a novel class of adenosine A1 receptor antagonists. Depending on ... Pyrazolo[3,4-b]pyridines have been recently presented as a novel class of adenosine A1 receptor antagonists. Depending on ... pyrimidine derivatives as antagonists for A1 adenosine receptor.. CICHERO, ELENA;CASOLINO, MARIA CHIARA;MENOZZI, GIULIA;MOSTI, ... In this work, we present a QSAR study on these analogues as antagonists for adenosine A1 receptors. Using the MOE software we ...
1,2,3-triazolo[5,4-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives: A new class of A(2A) adenosine receptor antagonists
... compared with A1 adenosine receptors.. 1,2,3-triazolo[5,4-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives: A new class of A(2A) ... adenosine receptor antagonists. BARALDI, Pier Giovanni;CACCIARI, Barbara;SPALLUTO G;PINEDA DE LAS INFANTAS MJ;ZOCCHI C;FERRARA ... were synthesized and tested as antagonists in receptor binding and in vitro functional assays to evaluate their potency for A( ... were synthesized and tested as antagonists in receptor binding and in vitro functional assays to evaluate their potency for A( ...
Gravidanza e allattamento
53) VAN DER GRAAF, P.H., SHANKLEY, N.P. & BLACK, J.W. (1996). Analysis of the activity of a1-adrenoceptor antagonists in rat ... 18) HAN, C. & MINNEMAN, K.P. (1991). Interaction of subtype-selective antagonist with a-adrenergic receptor binding sites in ... Effects of plant extract neferine on cyclic adenosine monophosphate and cyclic guanosine monophosphate levels in rabbit corpus ... Molecular cloning and expression of the cDNA for the hamster a1-adrenergic receptor. Proc. Natl. Acad. Sci. U.S.A., 85, 7159- ...